Document Type

Article

Publication Date

10-1-1999

Publication Title

Tetrahedron Letters

Volume

55

Issue

40

Publisher Name

Elsevier

Abstract

A racemic synthesis of azanoradamantane (±)-3 was accomplished via Yamamoto's MAD-catalyzed Diels-Alder protocol. Subsequently, a scalable asymmetric synthesis of azanoradamantane benzamide SC-52491 was carried out employing Helmchen's asymmetric Diels-Alder methodology to construct all four contiguous asymmetric centers with the correct relative stereochemistry and in 99.3% e.e.

Comments

Author Posting © Elsevier, 1999. This is the author's version of the work. It is posted here by permission of Elsevier for personal use, not for redistribution. The definitive version was published in Tetrahedron, Volume 55, Issue 40, October 1, 1999. http://dx.doi.org/10.1016/S0040-4020(99)00680-8

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This work is licensed under a Creative Commons Attribution-Noncommercial-No Derivative Works 3.0 License.

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